نتایج جستجو برای: alkylthio imidazole derivatives

تعداد نتایج: 111131  

2003
Weidong Zhang

Nucleophilic carbenes have recently emerged as powerful 1,1-dipole equivalents for the construction of functionalized hydroindolone derivatives via a novel [4+1] cycloaddition with vinyl isocyanates in our laboratory. This methodology has been successfully used in the total synthesis of several alkaloids, such as tazettine and mesembrine. Currently, we are investigating the total synthesis of s...

2014
RANGASWAMY ROOPASHREE CHAKRABHAVI DHANANJAYA MOHAN TORESHETTAHALLY RAMESH SWAROOP SWAMY JAGADISH

Objective: Cancer is one of the major causes of death worldwide irrespective of the sex. The aim of the study was to design, synthesize, and identification of novel anti-proliferative agents that can potently target cancer. Methods: We are reporting the synthesis of the new series of N-substituted 2-(2-butyl-4-chloro-1H-imidazole-5-yl)-1H-benzo[d]imidazole derivatives and evaluated for their an...

Journal: :Molecules 2013
Karlo Wittine Kristina Poljak Matea Kovač Damjan Makuc Janez Plavec Jan Balzarini Tamara Martinović Sandra Kraljević Pavelić Krešimir Pavelić Mladen Mintas

In the present paper, we report on the synthesis, and in vitro antiviral and cytostatic activities of a series of novel imidazole[4,5-e][1,3]diazepine-4,8-dione (compounds 9-11) and acyclic carbamoyl imino-ureido imidazole (compounds 12 and 13) derivatives. These new type of chemical entities showed no significant activity on the broad spectrum of DNA and RNA viruses. Results of antiproliferati...

Journal: :Chemical & pharmaceutical bulletin 2000
K Hori A Sakaguchi M Kudoh K Ishida Y Aoyama Y Yoshida

Fungicidal activity of widely used imidazole antifungal drugs in topical applications is not so strong in spite of their fungistatic activities against dermatophytes and pathogenic yeasts. In order to improve fungicidal activity of imidazole antifungal agents, a series of novel imidazole derivatives having a hydrophobic substituent derived from isoprenoid were synthesized. The efficacy of these...

Journal: :Indian Journal of Pharmaceutical and Biological Research 2017

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