نتایج جستجو برای: 5α dihydrotestosterone

تعداد نتایج: 3573  

Journal: :American journal of physiology. Endocrinology and metabolism 2014
Stephen E Borst Joshua F Yarrow Christine F Conover Unyime Nseyo John R Meuleman Judyta A Lipinska Randy W Braith Darren T Beck Jeffrey S Martin Matthew Morrow Shirley Roessner Luke A Beggs Sean C McCoy Darryl F Cannady Jonathan J Shuster

Testosterone acts directly at androgen receptors and also exerts potent actions following 5α-reduction to dihydrotestosterone (DHT). Finasteride (type II 5α-reductase inhibitor) lowers DHT and is used to treat benign prostatic hyperplasia. However, it is unknown whether elevated DHT mediates either beneficial musculoskeletal effects or prostate enlargement resulting from higher-than-replacement...

2012
Alicia A. Walf Cheryl A. Frye

Stressors, during early life or adulthood, can alter steroid-sensitive behaviors, such as exploration, anxiety, and/or cognitive processes. We investigated if exposure to acute stressors in adulthood may alter behavioral and neuroendocrine responses of male rats that were exposed to gestational stress or not. We hypothesized that rats exposed to gestational and acute stress may show behavioral ...

2014
Rita Upreti Katherine A. Hughes Dawn E. W. Livingstone Calum D. Gray Fiona C. Minns David P. Macfarlane Ian Marshall Laurence H. Stewart Brian R. Walker Ruth Andrew

CONTEXT 5α-Reductase (5αR) types 1 and 2 catalyze the A-ring reduction of steroids, including androgens and glucocorticoids. 5α-R inhibitors lower dihydrotestosterone in benign prostatic hyperplasia; finasteride inhibits 5αR2, and dutasteride inhibits both 5αR2 and 5αR1. In rodents, loss of 5αR1 promotes fatty liver. OBJECTIVE Our objective was to test the hypothesis that inhibition of 5αR1 c...

2015
Michela Di Mauro Alessandro Tozzi Paolo Calabresi Vito Enrico Pettorossi Silvarosa Grassi

Estrogenic and androgenic steroids synthesized in the brain may rapidly modulate synaptic plasticity interacting with specific membrane receptors. We explored by electrophysiological recordings in hippocampal slices of male rat the influence of 17β-estradiol (E2) and 5α-dihydrotestosterone (DHT) neo-synthesis on the synaptic changes induced in the CA1 region. Induction of long-term depression (...

2014
JOHN M. LACY NATASHA KYPRIANOU

The use of 5α-reductase inhibitors (5α-RIs) as prostate cancer chemoprevention agents is controversial. Two large randomized trials, the Prostate Cancer Prevention Trial (PCPT) and the Reduction by Dutasteride of Prostate Cancer Events (REDUCE) Trial, have both shown a decreased incidence of prostate cancer in patients administered with 5α-RIs. Both studies showed, however, an increased risk of...

2012
Michael G. Zager Hugh A. Barton

A systems-level mathematical model is presented that describes the effects of inhibiting the enzyme 5α-reductase (5aR) on the ventral prostate of the adult male rat under chronic administration of the 5aR inhibitor, finasteride. 5aR is essential for androgen regulation in males, both in normal conditions and disease states. The hormone kinetics and downstream effects on reproductive organs asso...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید