نتایج جستجو برای: tetralin

تعداد نتایج: 446  

Journal: :The Journal of pharmacology and experimental therapeutics 2003
Lalitha Madhavan William J Freed Vellareddy Anantharam Anumantha G Kanthasamy

Apoptosis and glutamate-mediated excitotoxicity may play a role in the pathogenesis of many neurodegenerative disorders, including Parkinson's disease (PD). In the present study, we investigated whether stimulation of the 5-hydroxytryptamine 1A (5-HT1A) receptor attenuates N-methyl-D-aspartate- (NMDA) and 1-methyl-4-phenylpyridinium (MPP(+))-induced apoptotic cell death in cell culture models. ...

Journal: :The Quarterly journal of experimental psychology. B, Comparative and physiological psychology 2000
H J Cassaday E L Simpson E A Gaffan

The 5-hydroxytryptamine1a (5-HT1a) receptor agonist 8-hydroxy-2-(di-n-propylamino) tetralin (8-OH-DPAT; 0.15 mg/kg) impaired rats' rapid visual learning on a computerized maze. This treatment also increased decision time (DT) but the learning impairment was not necessarily a side-effect of slower responding because, in this task, responses made at long DT are more accurate than those at short D...

Journal: :The Journal of pharmacology and experimental therapeutics 1997
L Johansson D Sohn S O Thorberg D M Jackson D Kelder L G Larsson L Rényi S B Ross C Wallsten H Eriksson P S Hu E Jerning N Mohell A Westlind-Danielsson

The pharmacological properties of a novel selective 5-hydroxytryptamine1A (5-HT1A) receptor antagonist, NAD-299 [(R)-3-N,N-dicyclobutylamino-8-fluoro-3,4-dihydro-2H-1-benzopyran-5-carboxamide hydrogen (2R,3R)-tartrate monohydrate] were examined in vitro and in vivo and compared with the reference 5-HT1A receptor antagonist, WAY-100635 [N-(2-(1-(4-(2-methoxyphenyl)piperazin-yl))ethyl)-N-(2-pyrid...

Journal: :Journal of medicinal chemistry 2011
Carmen Abate Mauro Niso Enza Lacivita Philip D Mosier Annamaria Toscano Roberto Perrone

1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine 1 (PB28) represents an excellent lead candidate for therapeutic and/or diagnostic applications in oncology. However, because its utility is limited by its relatively high degree of lipophilicity, novel analogues of 1 with reduced lipophilic character were designed by substituting methylene groups with more polar fu...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید