نتایج جستجو برای: n cyclohexyl 2

تعداد نتایج: 3133276  

Journal: :The Journal of pharmacology and experimental therapeutics 2009
Cynthia M Rominger Wei-Lin Tiger Bee Robert A Copeland Elizabeth A Davenport Aidan Gilmartin Richard Gontarek Keith R Hornberger Lorena A Kallal Zhihong Lai Kenneth Lawrie Quinn Lu Lynette McMillan Maggie Truong Peter J Tummino Brandon Turunen Matthew Will William J Zuercher David H Rominger

The Smoothened receptor (Smo) mediates hedgehog (Hh) signaling critical for development, cell growth, and migration, as well as stem cell maintenance. Aberrant Hh signaling pathway activation has been implicated in a variety of cancers, and small-molecule antagonists of Smo have entered human clinical trials for the treatment of cancer. Here, we report the biochemical characterization of allost...

Journal: :Journal of pharmaceutical sciences 1978
I Bartosek S Daniel S Sýkora

A polarographic method was developed to determine the antineoplastic agent carmustine and other nitrosoureas, such as N-methyl-N-nitrosourea and N-cyclohexyl-N-nitrosourea, in biological fluids at levels well below 1 microgram/ml or g. The stability of carmustine in different media was investigated to prevent losses during administration or assay. Examples of nitrosourea determination in biolog...

Journal: :Acta Crystallographica Section E Structure Reports Online 2012

Journal: :Molecules 2015
Tiago Fernandes da Silva Walfrido Bispo Júnior Magna Suzana Alexandre-Moreira Fanny Nascimento Costa Carlos Eduardo da Silva Monteiro Fabio Furlan Ferreira Regina Cely Rodrigues Barroso François Noël Roberto Takashi Sudo Gisele Zapata-Sudo Lídia Moreira Lima Eliezer J Barreiro

The N-acylhydrazone (NAH) moiety is considered a privileged structure, being present in many compounds with diverse pharmacological activities. Among the activities attributed to NAH derivatives anti-inflammatory and analgesic ones are recurrent. As part of a research program aiming at the design of new analgesic and anti-inflammatory lead-candidates, a series of cyclohexyl-N-acylhydrazones 10-...

Journal: :Organic & biomolecular chemistry 2008
Graham Stones Régis Tripoli Colin L McDavid Kewin Roux-Duplâtre Alan R Kennedy David C Sherrington Colin L Gibson

Two routes to the synthesis of a cyclohexyl-fused 1,4,7-triazacyclononane involving macrocyclisations of tosamides have been investigated. In the first approach, using a classic Richman-Atkins-type cyclisation of a cyclohexyl-substituted 1,4,7-tritosamide with ethylene glycol ditosylate, afforded the cyclohexyl-fused 1,4,7-triazacyclononane in 5.86% overall yield in four steps. The second, more...

Journal: :Acta Crystallographica Section E Structure Reports Online 2014

Journal: :Journal of Polymer Science Part A: General Papers 1965

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