نتایج جستجو برای: huperzine a

تعداد نتایج: 13431799  

Journal: :Epilepsy Research 2002
Meir Bialer Svein I. Johannessen René H. Levy Emilio Perucca Torbjörn Tomson H. Steve White

The Eigth Eilat Conference on New Antiepileptic Drugs (AEDs)-EILAT VII, took place in Sitges, Barcelona from the 10th to 14th September, 2006. Basic scientists, clinical pharmacologists and neurologists from 24 countries attended the conference, whose main themes included a focus on status epilepticus (epidemiology, current and future treatments), evidence-based treatment guidelines and the pot...

Journal: :Molecules 2017
Eva Mezeiova Jan Korabecny Vendula Sepsova Martina Hrabinova Petr Jost Lubica Muckova Tomas Kucera Rafael Dolezal Jan Misik Katarina Spilovska Ngoc Lam Pham Lucia Pokrievkova Jaroslav Roh Daniel Jun Ondrej Soukup Daniel Kaping Kamil Kuca

Tacrine (THA), the first clinically effective acetylcholinesterase (AChE) inhibitor and the first approved drug for the treatment of Alzheimer's disease (AD), was withdrawn from the market due to its side effects, particularly its hepatotoxicity. Nowadays, THA serves as a valuable scaffold for the design of novel agents potentially applicable for AD treatment. One such compound, namely 7-methox...

Journal: :Zhongguo yao li xue bao = Acta pharmacologica Sinica 1997
J H Lin G Y Hu X C Tang

AIM To compare the effects of huperzine A (Hup A), tacrine, and E2020 on cholinergic transmission at mouse neuromuscular junction in vitro. METHODS The isolated mouse phrenic nerve-hemidiaphragm preparations were used with the conventional intracellular recording technique. The miniature end-plate potentials (MEPP), the mean quantal content of end-plate potentials (EPP), and the resting membr...

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