نتایج جستجو برای: antiplasmodial activity

تعداد نتایج: 1134718  

Journal: :PLoS pathogens 2018
Erick T Tjhin Christina Spry Alan L Sewell Annabelle Hoegl Leanne Barnard Anna E Sexton Ghizal Siddiqui Vanessa M Howieson Alexander G Maier Darren J Creek Erick Strauss Rodolfo Marquez Karine Auclair Kevin J Saliba

The malaria-causing blood stage of Plasmodium falciparum requires extracellular pantothenate for proliferation. The parasite converts pantothenate into coenzyme A (CoA) via five enzymes, the first being a pantothenate kinase (PfPanK). Multiple antiplasmodial pantothenate analogues, including pantothenol and CJ-15,801, kill the parasite by targeting CoA biosynthesis/utilisation. Their mechanism ...

Journal: :Molecules 2017
Tawanda Zininga Lebogang Ramatsui Pertunia Bveledzani Makhado Stanley Makumire Ikechukwu Achilinou Heinrich Hoppe Heini Dirr Addmore Shonhai

Heat shock proteins (Hsps), amongst them, Hsp70 and Hsp90 families, serve mainly as facilitators of protein folding (molecular chaperones) of the cell. The Hsp70 family of proteins represents one of the most important molecular chaperones in the cell. Plasmodium falciparum, the main agent of malaria, expresses six Hsp70 isoforms. Two (PfHsp70-1 and PfHsp70-z) of these localize to the parasite c...

2014
Vincent E. Rasamison L. Harinantenaina Rakotondraibe Carla Slebodnick Peggy J. Brodie Michel Ratsimbason Karen TenDyke Yongchun Shen Lucien M. Randrianjanaka David G. I. Kingston

The new triterpene turranoic acid (1) and the new N-containing nor-triterpene turraenine (2), along with triptocallic acid B (3) and esculentoic acid (4) were isolated from leaves of a Turraea sp. Compounds 1-3 showed weak to moderate in vitro antiplasmodial activity against the chloroquine-resistant Plasmodium falciparum strain FCM29. Compound 1 also displayed weak cytotoxic activity against t...

Journal: :Tropical Medicine and International Health 1999

Journal: :Journal of Drug Delivery and Therapeutics 2023

Background: Despite the various medicinal applications of Schumanniophyton magnificum, no comparative data are available to determine part with best antiplasmodial activity and guarantee its safety. This work deals evaluation methanolic extracts S. magnificum organs as well study acute toxicity most active part.
 Materials methods: The leaves, stem bark, trunk wood, root wood were obtained...

Journal: :European journal of pharmacology 2006
Geneviève Philippe Laurent Nguyen Luc Angenot Michel Frédérich Gustave Moonen Monique Tits Jean-Michel Rigo

Strychnos icaja Baill. (Loganiaceae) is a liana found in Central Africa known to be an arrow and ordeal poison but also used by traditional medicine to treat malaria. Recently, many dimeric or trimeric indolomonoterpenic alkaloids with antiplasmodial properties have been isolated from its rootbark. Since these alkaloids are derivatives of strychnine, it was important, in view of their potential...

Journal: :Journal of ethnopharmacology 2012
Phurpa Wangchuk Paul A Keller Stephen G Pyne Anthony C Willis Sumalee Kamchonwongpaisan

ETHNOPHARMACOLOGICAL RELEVANCE Corydalis dubia is used in Bhutanese traditional medicine as a febrifuge and for treating infections in the blood, liver and bile which correlate to the signs and symptoms of malarial and microbial infections. AIM OF THE STUDY To validate the ethnopharmacological uses of the plant and to discover potential new therapeutic drug leads. MATERIALS AND METHODS C. d...

Journal: :Molecules 2013
Hsing-Tan Li Hui-Ming Wu Hsin-Liang Chen Chi-Ming Liu Chung-Yi Chen

Several species of Magnoliaceae and Annonaceae are used in Traditional Chinese Medicine. (-)-Anonaine, isolated from several species of Magnoliaceae and Annonaceae, presents antiplasmodial, antibacterial, antifungal, antioxidation, anticancer, antidepression, and vasorelaxant activity. This article provides an overview of the pharmacological functions of (-)-anonaine.

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