نتایج جستجو برای: 5 fluorouracil 5 fu

تعداد نتایج: 1223700  

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2011
Praveen K Nambaru Tobias Hübner Kathleen Köck Steffen Mews Markus Grube Léa Payen Jérôme Guitton Matthias Sendler Gabriele Jedlitschky Christian Rimmbach Dieter Rosskopf Dariusz W Kowalczyk Heyo K Kroemer Frank U Weiss Julia Mayerle Markus M Lerch Christoph A Ritter

Pancreatic adenocarcinoma is one of the malignancies that is highly resistant to therapy and among the leading causes of cancer-related death. Several factors may influence pancreatic cancer resistance, and expression of ATP-binding cassette transport proteins is one of the major mechanisms of drug resistance. Members of this family's C-branch, also referred to as multidrug resistance-associate...

2017
Masakazu Fukushima Kenzo Iizuka Cheng Jin Chun Zhang Mei Hong Kiyoshi Eshima

To reduce 5-fluorouracil (5-FU)-induced serious toxicities without loss of antitumor activity, we have developed DFP-11207, a novel fluoropyrimidine, which consists of 1-ethoxymethyl-5-fluorouracil (EM-FU; a precursor form of 5-FU), 5-chloro-2,4-dihydroxypyridine (CDHP; an inhibitor of 5-FU degradation), and citrazinic acid (CTA; an inhibitor of 5-FU phosphorylation). In vitro studies of DFP-11...

2011
Shuji Komori Shinji Osada Kazuhiro Yoshida

5-fluorouracil (5-FU) is widely used in chemotherapy for gastric and colorectal cancer, but gemcitabine (GEM), and not 5-FU, is approved as a standard drug for use in pancreatic cancer. Interindividual variation in the enzyme activity of the GEM metabolic pathway can affect the extent of GEM metabolism and the efficacy of GEM chemotherapy. Human equilibrative nucleoside transporter 1 (hENT1) is...

2009
In Jeong Cho Hye Jung Chang Kyoung Eun Lee Hye Sung Won Moon Young Choi Eun Mi Nam Yeung-Chul Mun Soon Nam Lee Chu-Myong Seong

The pyrimidine antimetabolite 5-fluorouracil (5-FU) is a chemotherapeutic agent used widely for various tumors. Common side effects of 5-FU are related to its effects on the bone marrow and gastrointestinal epithelium. Neurotoxicity caused by 5-FU is uncommon, although acute and delayed forms have been reported. Wernicke's encephalopathy is an acute, neuropsychiatric syndrome resulting from thi...

Journal: :International journal of pharmaceutics 2002
B Arica S Caliş H Kaş M Sargon A Hincal

Alginate beads containing 5-fluorouracil (5-FU) were prepared by the gelation of alginate with calcium cations. Alginate beads loaded with 5-FU were prepared at 1.0 and 2.0% (w/v) polymers. The effect of polymer concentration and the drug loading (1.0, 5.0 and 10%) on the release profile of 5-FU was investigated. As the drug load increased, larger beads were obtained in which the resultant bead...

2017
Samideh Khoei Roghayeh Poorabdollahi Ahmad Mostaar Fariborz Faeghi

OBJECTIVE This study intended to observe the effects of methoxyamine (Mx) on cytotoxic effects and DNA damage caused by 5-Fluorouracil (5-FU) in combination with gamma radiation in a human colon cancer cell line, HT29. MATERIALS AND METHODS In this experimental study, HT29 cells were cultured as a monolayer and treated with different concentrations of 5-FU along with 1 mM Mx for 24 hours. Nex...

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