نتایج جستجو برای: n amino 2 pyridones

تعداد نتایج: 3257200  

Journal: :Bioorganic & medicinal chemistry letters 2011
José M Bueno Pilar Manzano María C García Jesús Chicharro Margarita Puente Milagros Lorenzo Adolfo García Santiago Ferrer Rubén M Gómez María T Fraile José L Lavandera José M Fiandor Jaume Vidal Esperanza Herreros Domingo Gargallo-Viola

Antimalarial 4-pyridones are a novel class of inhibitors of the plasmodial mitochondrial electron transport chain targeting Cytochrome bc1 (complex III). In general, the most potent 4-pyridones are lipophilic molecules with poor solubility in aqueous media and low oral bioavailability in pre-clinical species from the solid dosage form. The strategy of introducing polar hydroxymethyl groups has ...

Journal: :Journal of Synthetic Organic Chemistry, Japan 2015

Journal: :Acta Crystallographica Section A Foundations and Advances 2017

Journal: :Acta Crystallographica Section E Structure Reports Online 2010

Journal: :Acta Crystallographica Section E Structure Reports Online 2009

2013
Yan-Hui Liang Xiang-Dong Mei Yao-Fa Li Wen-Liang Pan Jun Ning

In the title compound, C8H9ClN2O, the dihedral angle between the benzene ring and the methyl-amide substituent is 68.39 (11)°. In the crystal, mol-ecules are linked by N-H⋯O hydrogen bonds, forming layers parallel to the ab plane.

2012
Shaaban K. Mohamed Goran A. Bogdanović Mehmet Akkurt Antar A. Abdelhamid Sabry H. H. Younes

In the title compound, C(18)H(21)N(3)O(3), the terminal phenyl rings make a dihedral angle of 86.3 (5)°. In the crystal, mol-ecules are linked by N-H⋯O hydrogen bonds into chains along [001], forming parallel C(4) and R(1) (2)(6) graph-set motifs.

2012
Zhong-Feng Shi Jia-Ming Li

The title Schiff base compound, C(14)H(12)N(4)O(3), displays an E conformation with respect to the C=N double bond [1.268 (3) Å]. The dihedral angle between the benzene rings is 3.2 (5)°, consistent with an essentially planar mol-ecule. In the crystal, N-H⋯O and N-H⋯N hydrogen bonds, as well as C-H⋯O inter-actions, link the mol-ecules into layers that stack along the c axis.

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