نتایج جستجو برای: tricyclic graph

تعداد نتایج: 201825  

Journal: :The Journal of pharmacology and experimental therapeutics 2015
Jennifer Lu Veronique Michaud Liliam Gabriela Guilarte Moya Fleur Gaudette Yat Hei Leung Jacques Turgeon

The organic anion transporting polypeptide 1A2 (OATP1A2), a membrane drug transporter expressed on important organs (such as the brain, kidney, and intestine) may be a key element in the disposition of drugs. Previous studies demonstrated that it could transport a broad spectrum of substrates, including endogenous molecules and clinically relevant drugs, such as several β-blockers and 3-hydroxy...

2005
Michael J. Owens

ackground: The use of antidepressants during pregnancy continues to garner considerable attention, though there are limited nvestigations that have sought to quantify fetal exposure. ethods: Maternal and umbilical cord sera were collected at delivery from ten women taking nortriptyline and seven taking lomipramine. Placental passage was calculated as the ratio of umbilical cord to maternal seru...

Journal: :Journal of the Brazilian Chemical Society 2015

2010
Subhodeep Sarker René Weissensteiner Ilka Steiner Harald H Sitte Gerhard F Ecker Michael Freissmuth Sonja Sucic

The structure of the bacterial leucine transporter from Aquifex aeolicus (LeuT(Aa)) has been used as a model for mammalian Na(+)/Cl(-)-dependent transporters, in particular the serotonin transporter (SERT). The crystal structure of LeuT(Aa) liganded to tricyclic antidepressants predicts simultaneous binding of inhibitor and substrate. This is incompatible with the mutually competitive inhibitio...

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