نتایج جستجو برای: n 5

تعداد نتایج: 2009355  

Journal: :Bioorganic & medicinal chemistry letters 2011
Hayden Matthews Marie Ranson Joel D A Tyndall Michael J Kelso

A known side-activity of the oral potassium-sparing diuretic drug amiloride is inhibition of the enzyme urokinase-type plasminogen activator (uPA, K(i)=7 μM), a promising anticancer target. Several studies have demonstrated significant antitumor/metastasis properties for amiloride in animal cancer models and it would appear that these arise, at least in part, through inhibition of uPA. Selectiv...

2012
V. Giansanti G. Santamaria A. Torriglia F. Aredia A.I. Scovassi G. Bottiroli A.C. Croce

HMA (5-(N,N-hexamethylene)amiloride), which belongs to a family of novel amiloride derivatives, is one of the most effective inhibitors of Na+/H+ exchangers, while uneffective against Na+ channels and Na+/Ca2+ exchangers. In this study, we provided evidence that HMA can act as a fluorescent probe. In fact, human retinal ARPE19 cells incubated with HMA show an intense bluish fluorescence in the ...

Journal: :Acta Crystallographica Section E Structure Reports Online 2011

Journal: :Acta Crystallographica Section E Structure Reports Online 2010

Journal: :Acta Crystallographica Section E Structure Reports Online 2010

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