نتایج جستجو برای: histamine h2 receptor

تعداد نتایج: 622815  

2006

A key role for histamine in the physiological control of gastric acid secretion was established with the advent of the histamine H2-receptor antagonists which have in vivo been shown to inhibit virtually all forms of basal and stimulated secretion.' These data can be seen to support the common mediator hypothesis championed in the last three decades by Code2 3 and which states that secretory st...

2006

A key role for histamine in the physiological control of gastric acid secretion was established with the advent of the histamine H2-receptor antagonists which have in vivo been shown to inhibit virtually all forms of basal and stimulated secretion.' These data can be seen to support the common mediator hypothesis championed in the last three decades by Code2 3 and which states that secretory st...

Journal: :The Journal of pharmacology and experimental therapeutics 2009
Hidenori Wake Hideo Kohka Takahashi Shuji Mori Keyue Liu Tadashi Yoshino Masahiro Nishibori

Advanced glycation end products (AGEs) are modifications of proteins/lipids that become nonenzymatically glycated after contact with aldose sugars. Among various subtypes of AGEs, glyceraldehyde-derived AGE (AGE-2) and glycolaldehyde-derived AGE (AGE-3) are suggested to play roles in inflammation in diabetic patients. Because the engagement of intercellular adhesion molecule (ICAM)-1, B7.1, B7....

E Tamaddonfard G Vafaye Saiah

Several lines of evidence suggest that brain histamine may be involved in the central control of food intake. The effect of histamine on feeding is mediated through three kinds of receptors (H1, H2, and H3). The present study was designed to investigate the effect of intracerebroventricular injection of histamine, promethazine (H1 antagonist) and ranitidine (H2 antagonist) on food intake of fre...

2014
Sang Eok Lee Dae Hoon Kim Young Chul Kim Joung-Ho Han Woong Choi Chan Hyung Kim Hye Won Jeong Seon-Mee Park Sei Jin Yun Song-Yi Choi Rohyun Sung Young Ho Kim Ra Young Yoo Park Hee Sun Heon Kim Young-Jin Song Wen-Xie Xu Hyo-Yung Yun Sang Jin Lee

This study was designed to examine the effects of histamine on gastric motility and its specific receptor in the circular smooth muscle of the human gastric corpus. Histamine mainly produced tonic relaxation in a concentration-dependent and reversible manner, although histamine enhanced contractility in a minor portion of tissues tested. Histamine-induced tonic relaxation was nerve-insensitive ...

Journal: :The American journal of physiology 1997
John Del Valle Ira Gantz

Histamine exerts multiple biological actions through one of three receptor subtypes (H1, H2, and H3). This review focuses on new developments regarding the structure and function of the H2 receptor. In addition to the important role this receptor plays in stimulating gastric acid secretion, recent studies have demonstrated that it is also involved in regulating gastrointestinal motility and int...

2013
Thomas K Pellinger Breanna R Dumke John R Halliwill

Following a bout of dynamic exercise, humans experience sustained postexercise vasodilatation in the previously exercised skeletal muscle which is mediated by activation of histamine (H1 and H2) receptors. Skeletal muscle glucose uptake is also enhanced following dynamic exercise. Our aim was to determine if blunting the vasodilatation during recovery from exercise would have an adverse effect ...

Journal: :The Yale Journal of Biology and Medicine 1992
N. P. Shankley N. J. Welsh J. W. Black

Does gastrin stimulate gastric acid secretion by direct action on oxyntic cells, by releasing histamine, or by being potentiated by histamine? Previous studies in the mouse pointed to gastrin-regulated histamine release. Guinea pig and rat are well known to vary in their sensitivity to histamine. Therefore, the effects of histamine and pentagastrin were compared quantitatively on isolated, lume...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2005
Fabio Cianchi Camillo Cortesini Nicola Schiavone Federico Perna Lucia Magnelli Elena Fanti Daniele Bani Luca Messerini Valentina Fabbroni Giuliano Perigli Sergio Capaccioli Emanuela Masini

PURPOSE Activity of histidine decarboxylase, the key enzyme in the synthesis of histamine, has been shown to be increased in several types of human tumors. We attempted to establish whether the possible involvement of histidine decarboxylase and histamine in colorectal carcinogenesis might be mediated by the activation of the cyclooxygenase-2 (COX-2) pathway. EXPERIMENTAL DESIGN Expression/ac...

2015
Robin L. Thurmond

The histamine H4 receptor (H4R) was first noted as a sequence in genomic databases that had features of a class A G-protein coupled receptor. This putative receptor was found to bind histamine consistent with its homology to other histamine receptors and thus became the fourth member of the histamine receptor family. Due to the previous success of drugs that target the H1 and H2 receptors, an e...

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