نتایج جستجو برای: small molecule

تعداد نتایج: 886075  

Journal: :ACS chemical biology 2016
Matthew D Disney Audrey M Winkelsas Sai Pradeep Velagapudi Mark Southern Mohammad Fallahi Jessica L Childs-Disney

The development of small molecules that target RNA is challenging yet, if successful, could advance the development of chemical probes to study RNA function or precision therapeutics to treat RNA-mediated disease. Previously, we described Inforna, an approach that can mine motifs (secondary structures) within target RNAs, which is deduced from the RNA sequence, and compare them to a database of...

2016
Nuha R. Mansour Ross Paveley J. Mark F. Gardner Andrew S. Bell Tanya Parkinson Quentin Bickle

An estimated 600 million people are affected by the helminth disease schistosomiasis caused by parasites of the genus Schistosoma. There is currently only one drug recommended for treating schistosomiasis, praziquantel (PZQ), which is effective against adult worms but not against the juvenile stage. In an attempt to identify improved drugs for treating the disease, we have carried out high thro...

Journal: :Bioorganic & medicinal chemistry 2015
Ignacio Colomer Ololade Adeniji George M Burslem Philip Craven Martin Ohsten Rasmussen Anthony Willaume Tuomo Kalliokoski Richard Foster Stephen P Marsden Adam Nelson

The application of [4+2] cycloadditions between alkenes and an N-benzoyl iminium species, generated in situ under acidic conditions, is described in the synthesis of diverse molecular scaffolds. The key reaction led to the formation of cyclic imidates in good yield and with high regioselectivity. It was demonstrated that the cyclic imidates may be readily converted into 1,3-amino alcohols. Inco...

Journal: :Molecular Systems Biology 2008

Journal: :Frontiers in Pharmacology 2020

Journal: :Chemistry & Biology 2010

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