نتایج جستجو برای: imidazoline

تعداد نتایج: 848  

Journal: :Journal of medicinal chemistry 1997
F Rondu G Le Bihan X Wang A Lamouri E Touboul G Dive T Bellahsene B Pfeiffer P Renard B Guardiola-Lemaitre D Manechez L Penicaud A Ktorza J J Godfroid

The physiopathology of non-insulin-dependent diabetes mellitus is associated with a dysfunction in the regulation of insulin secretion. The alpha 2-adrenoceptors have been reported to be involved in this alteration, although alpha 2-antagonists containing an imidazoline ring may stimulate insulin secretion independently of alpha 2-adrenoceptor blockage. Recently, a new "imidazoline-binding site...

Journal: :The Journal of pharmacology and experimental therapeutics 2004
Rouwayda El-Ayoubi Ahmed Menaouar Jolanta Gutkowska Suhayla Mukaddam-Daher

We have recently identified imidazoline I(1)-receptors in the heart. In the present study, we tested regulation of cardiac I(1)-receptors versus alpha(2) -adrenoceptors in response to hypertension and to chronic exposure to agonist. Spontaneously hypertensive rats (SHR, 12-14 weeks old) received moxonidine (10, 60, and 120 microg/kg/h s.c.) for 1 and 4 weeks. Autoradiographic binding of (125)I-...

2008
Jiu Li Chang Zhi Yong Gao Kai Jiang

The title compound C(12)H(17)N(3)O(2) (+)·Cl(-) consists of a discrete [NITpPyH](+) cation [NITpPy = 2-(4'-pyrid-yl)-4,4,5,5-tetra-methyl-imidazoline-1-oxyl-3-oxide] and a chloride anion. The NITpPy mol-ecule is protonated at the N atom of the pyridyl ring. The anions and cations are connected via N-H⋯Cl hydrogen bonds.

Journal: :Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 1997
K Kalantar-Zadeh K Singh M Kleiner M P Jarrett F C Luft

Key words: patellar tendon; bilateral tendon rupture; lems were reported. Her current medications included chronic renal failure; secondary hyperparathyroidism; an angiotensin converting enzyme inhibitor, a long-haemarthrosis acting calcium channel blocker, a centrally acting imidazoline derivative, and famotidine. Ferrous sulfate and subcutaneous recombinant human erythropoietin were given for...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 2007
Mahesh S Joshi T Bruce Ferguson Fruzsina K Johnson Robert A Johnson Sampath Parthasarathy Jack R Lancaster

Arginine contains the guanidinium group and thus has structural similarity to ligands of imidazoline and alpha-2 adrenoceptors (alpha-2 AR). Therefore, we investigated the possibility that exogenous arginine may act as a ligand for these receptors in human umbilical vein endothelial cells and activate intracellular nitric oxide (NO) synthesis. Idazoxan, a mixed antagonist of imidazoline and alp...

Journal: :The Journal of pharmacology and experimental therapeutics 2000
R Raddatz S L Savic V Bakthavachalam J Lesnick J R Jasper C R McGrath A Parini S M Lanier

A series of phenoxy-substituted methylimidazoline derivatives were synthesized and used to define the ligand recognition properties of the imidazoline-binding domain (IBD) on monoamine oxidase (MAO)-B and its role in substrate processing. The rank order of potency for selected compounds in competitive binding studies with the imidazoline [(3)H]idazoxan was different from that in enzyme activity...

2010
Hoong-Kun Fun Jia Hao Goh Arnab Kar Shyamaprosad Goswami

In the title compound, guanidinium chloridotrioxidochrom-ate(VI), (CH(6)N(3))[CrClO(3)], both the cation and anion are generated by crystallographic mirror symmetry, with one O and one N atom and the Cr, Cl and C atoms lying on the mirror plane. The bond lengths in the guanidinium cation are inter-mediate between normal C-N and C=N bond lengths, indicating significant delocalization in this spe...

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