نتایج جستجو برای: antimalarial

تعداد نتایج: 6488  

Journal: :Bioorganic & medicinal chemistry 2004
Dora Carrico Junko Ohkanda Howard Kendrick Kohei Yokoyama Michelle A Blaskovich Cynthia J Bucher Frederick S Buckner Wesley C Van Voorhis Debopam Chakrabarti Simon L Croft Michael H Gelb Saïd M Sebti Andrew D Hamilton

A series of protein farnesyltransferase inhibitor ester prodrugs of FTI-2148 (17) were synthesized in order to evaluate the effects of ester structure modification on antimalarial activity and for further development of a farnesyltransferase inhibitor with in vivo activity. Evaluation against P. falciparum in red blood cells showed that all the investigated esters exhibited significant antimala...

Journal: :Experimental parasitology 2011
C N Muthaura J M Keriko S Derese A Yenesew G M Rukunga

Malaria is a major public health problem in many tropical and subtropical countries and the burden of this disease is getting worse, mainly due to the increasing resistance of Plasmodium falciparum against the widely available antimalarial drugs. There is an urgent need for discovery of new antimalarial agents. Herbal medicines for the treatment of various diseases including malaria are an impo...

Journal: :The Journal of antimicrobial chemotherapy 2006
Alexis Nzila

Chemotherapy remains the most important means of controlling malaria, one of the deadliest infectious parasitic diseases in the world. Antimalarial antifolates have been central for prophylaxis and treatment of malaria. This drug family was discovered in the 1940s, during the Second World War, and molecules that are currently in clinical use were discovered at that time. Since the 1940s, no new...

2016
Rosemin Kassam Richard Sekiwunga John B Collins Juliet Tembe Eric Liow

BACKGROUND This study responds to a rural community's concern that, despite national initiatives, malaria management in young children falls short of national guidelines in their district. This study aimed to: (1) describe caregivers' treatment-seeking behaviors in the rural district of Butaleja, (2) estimate the percentage of children who received an appropriate antimalarial, and (3) determine...

Journal: :British medical journal 1982
K M De Cock

The incidence of cases of malaria imported into the United Kingdom has increased.1 2 Early and appropriate treatment in Steroid-dependent patients are vulnerable to severe cases is vital, but hospital pharmacies may not always overwhelming infection with falciparum malaria stock parenteral antimalarial drugs. We report-on a case of fatal and other parasites. Parenteral antimalarial falciparum m...

Journal: :Journal of Clinical Investigation 2004

اسدالهی, اقباله, اونیل, پروفسور پال, خسروی, افرا,

Background and Objective: Resistance to chloroquine (CQ) in Plasmodium falciparum malaria has become a major health concern in the developing countries. This problem has prompted investigators for finding alternative antimalarials that may be effective against resistant strains. Amodiaquine (AQ) is an antimalarial which is effective against many chloroquine-resistant strains of P. falciparum. H...

Scrophularia umbrosa is a medicinal plant used as a traditional herb. This study was designed to investigate the phytochemical analysis of methanol (MeOH), DCM, and n-Hexane extracts of rhizome as well as total phenol and total flavonoid contents (TPC and TFC). In-vitro β-hematin formation assay and DPPH method were applied for analyzing antimalarial and free-radical scavenging activities of th...

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