Palladium-catalyzed direct and regioselective C-H acyloxylation of indolizines.
نویسندگان
چکیده
A direct and regioselective C1-acyloxylation of indolizines was developed via palladium-catalyzed C-H functionalization. A series of indolizines were successfully acyloxylated at the C1 position with the tolerance of a broad range of functional groups. In this reaction, high regioselectivity was achieved in the absence of a directing group. This work represents the first example of indolizine acyloxylation via C-H activation.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 13 40 شماره
صفحات -
تاریخ انتشار 2015